BTK gatekeeper residue variation combined with cysteine 481 substitution causes super-resistance to irreversible inhibitors acalabrutinib, ibrutinib and zanubrutinib
In: Leukemia, Jg. 35 (2021), Heft 8, S. 1317-1329
Online
academicJournal
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BTK gatekeeper residue variation combined with cysteine 481 substitution causes super-resistance to irreversible inhibitors acalabrutinib, ibrutinib and zanubrutinib
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Autor/in / Beteiligte Person: | Estupinan, HY ; Wang, Q ; Berglof, A ; Schaafsma, GCP ; Shi, YY ; Zhou, LT ; Mohammad, DK ; Yu, L ; Vihinen, M ; Zain, R ; Smith, CIE |
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Zeitschrift: | Leukemia, Jg. 35 (2021), Heft 8, S. 1317-1329 |
Veröffentlichung: | 2021 |
Medientyp: | academicJournal |
ISSN: | 1476-5551 (print) |
DOI: | 10.1038/s41375-021-01123-6 |
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